Published November 1992 | Version v1
Journal article

Study of the distribution and kinetics of [14C] sarcolysine in rats

  • 1. N.N. Petrov Scientific-Research Institute of Oncology, Leningrad (Russian Federation)

Description

One of the first antitumor drugs -- sarcolysine [4-bis(2-chloroethyl)-aminophenylalanine, mixture of isomers] and its L-isomer, melfalan, have been widely used clinically up to this time. A number of researchers have used various methods to study the pharmocokinetics of the drug in rats, mice, rabbits, dogs, monkeys, and humans. The aim of the present investigation was to study the complex of kinetic parameters of sarcolysine in rats in the case of various modes of administration and doses. The studies were conducted on noninbred white rats using [14C]sarcolysine. 12 refs., 2 figs., 2 tabs

Additional details

Publishing Information

Journal Title
Pharmaceutical Chemistry Journal
Journal Volume
26
Journal Issue
1
Journal Page Range
p. 30-33.
ISSN
0091-150X
CODEN
PCJOAU

INIS

Country of Publication
United States
Country of Input or Organization
United States
INIS RN
25014919
Subject category
S62: RADIOLOGY AND NUCLEAR MEDICINE;
Resource subtype / Literary indicator
Translation
Descriptors DEI
ANTINEOPLASTIC DRUGS; CARBON 14 COMPOUNDS; DOSE-RESPONSE RELATIONSHIPS; ISOMERS; LABELLING; METABOLISM; PHARMACOLOGY; RADIONUCLIDE ADMINISTRATION; RADIONUCLIDE KINETICS; RATS; TISSUE DISTRIBUTION
Descriptors DEC
ANIMALS; CARBON COMPOUNDS; DISTRIBUTION; DRUGS; KINETICS; MAMMALS; RODENTS; VERTEBRATES

Optional Information

Notes
Translated from Khimiko-farmatsevticheskii Zhurnal; 26: No. 1, 25-27(Jan 1992).