Published August 1987 | Version v1
Journal article

Synthesis of [3-3H]-4β, 15-diacetoxy-8α-(3-methylbutyryloxy)-3α-hydroxy-12, 13-epoxytrichothec-9-ene

  • 1. Academy of Military Medical Sciences, PLA, Beijing (China). Inst. of Pharmacology and Toxicology
  • 2. Academia Sinica, Beijing, BJ (China). Inst. of Atomic Energy

Description

[3-3H]-4β, 15-diacetoxy-8α-(3-methylburyloxy)-3α-hydroxy-12, 13-epoxy trichothec-9-ene is synthetized by oxidizing the C-3-hydroxy to ketone. It is reduced with NaB3H4 to a mixture of epimers which are separable by high thin-layer chromatography. The sepcific activity is 629 GBq/mmol and radiochemical purity is over 98%. Specific activity of this tritium labeled T-2-toxin is higher than that by Wallace

Additional details

Publishing Information

Journal Title
J. Nucl. Radiochem.
Journal Volume
9
Journal Issue
3
Series
J. Nucl. Radiochem.
Journal Page Range
190-192
ISSN
0253-9950
CODEN
HHHHD