Published February 8, 2000 | Version v1
Patent

Rigid bifunctional chelating agents

Description

Bicyclo[2.2.2]octane-2,3 diamine-N,N,N,Nprime-tetraacetic acids (BODTA) and bicyclo[2.2.1]heptane-2,3 diamine-N,N,Nprime,Nprime-tetraacetic acid (BHDTA) are chelating agents useful in forming detectably labeled bioconjugate compounds for diagnostic and therapeutic purposes. New compounds and processes of forming BODTA and BHDTA are disclosed. Radioimmunoconjugates of the present invention show high and prolonged tumor uptake with low normal tissue uptakes

Availability note (English)

Available from Patent and Trademark Office, Box 9, Washington, DC 20232 (US)

Additional details

Publishing Information

Imprint Pagination
[10 p.]
IPC:
Int. Cl. A61K 51/00; A61M 36/14
IPC
Int. Cl. A61K 51/00; A61M 36/14
Patent number
US patent document 9-046,030

INIS

Country of Publication
United States
Country of Input or Organization
United States
INIS RN
31024808
Subject category
S62: RADIOLOGY AND NUCLEAR MEDICINE;
Resource subtype / Literary indicator
Non-conventional Literature
Descriptors DEI
CHELATING AGENTS; DIAGNOSIS; NEOPLASMS; RADIOPHARMACEUTICALS; THERAPY; USES
Descriptors DEC
DISEASES; DRUGS; LABELLED COMPOUNDS; MATERIALS; MEDICINE; RADIOACTIVE MATERIALS

Optional Information

Notes
AC02-76CH00016
Secondary number(s)
US patent application 9-046,030