Published September 1996 | Version v1
Journal article Metadata-only

Synthesis of a carbon-14 labelled version of benzofuran GR151004B

Creators

  • 1. Glaxo Wellcome Research and Development, Isotope Chemistry Unit, Stevenage (United Kingdom)

Description

The 5HT1 receptor agonist GR151004B, labelled with carbon-14 at C-3 of the benzofuran ring, was prepared in 19% overall yield in five steps from 5-bromo-2-methoxybenzoic [14C]acid. (author)

Additional details

Publishing Information

Journal Title
Journal of Labelled Compounds and Radiopharmaceuticals
Journal Volume
38
Journal Issue
9
Journal Page Range
p. 863-871.
ISSN
0362-4803
CODEN
JLCRD4

INIS

Country of Publication
United Kingdom
Country of Input or Organization
United Kingdom
INIS RN
29007183
Subject category
S38: RADIATION CHEMISTRY, RADIOCHEMISTRY AND NUCLEAR CHEMISTRY;
Descriptors DEI
BENZOFURANS; CARBON 14 COMPOUNDS; CHEMICAL PREPARATION; LABELLING; RADIOPHARMACEUTICALS; RECEPTORS; SEROTONIN
Descriptors DEC
AMINES; AROMATICS; AUTONOMIC NERVOUS SYSTEM AGENTS; AZAARENES; AZOLES; CARBON COMPOUNDS; DRUGS; FURANS; HETEROCYCLIC COMPOUNDS; HYDROXY COMPOUNDS; INDOLES; LABELLED COMPOUNDS; MATERIALS; NEUROREGULATORS; ORGANIC COMPOUNDS; ORGANIC NITROGEN COMPOUNDS; ORGANIC OXYGEN COMPOUNDS; PYRROLES; RADIOACTIVE MATERIALS; RADIOPROTECTIVE SUBSTANCES; RESPONSE MODIFYING FACTORS; SYMPATHOMIMETICS; SYNTHESIS; TRYPTAMINES