Published July 1985 | Version v1
Journal article

Synthesis of (2R)- and (2S)-[3-2H]-valine

  • 1. Canterbury Univ., Christchurch (New Zealand). Dept. of Chemistry

Description

(2R)-Valine and the (2S)-isomer were esterified and benzoylated. The derivatives were chlorinated at C-3 by treatment with sulphuryl chloride, reduced to the 3-2H derivatives by reaction with triphenyltin deuteride, then hydrolysed to give (2R)- and (2S)-[3-2H]-valine. The labelling is achieved with complete retention of optical purity. (author)

Additional details

Publishing Information

Journal Title
J. Labelled Compd. Radiopharm.
Journal Volume
22
Journal Issue
7
Series
J. Labelled Compd. Radiopharm.
Journal Page Range
667-672
ISSN
0362-4803
CODEN
JLCRD

INIS

Country of Publication
United Kingdom
Country of Input or Organization
United Kingdom
INIS RN
17012006
Subject category
S37: INORGANIC, ORGANIC, PHYSICAL AND ANALYTICAL CHEMISTRY;
Descriptors DEI
CHEMICAL PREPARATION; DEUTERIUM COMPOUNDS; ISOMERS; LABELLING; VALINE
Descriptors DEC
AMINO ACIDS; CARBOXYLIC ACIDS; HYDROGEN COMPOUNDS; ORGANIC ACIDS; ORGANIC COMPOUNDS; SYNTHESIS